| CryptoSite: expanding the druggable proteome by characterization and prediction of cryptic binding sites P Cimermancic, P Weinkam, TJ Rettenmaier, L Bichmann, DA Keedy, ... Journal of molecular biology 428 (4), 709-719, 2016 | 211 | 2016 |
| Hydride as a leaving group in the reaction of pinacolborane with halides under ambient grignard and barbier conditions. One-Pot synthesis of alkyl, aryl, heteroaryl, vinyl, and … JW Clary, TJ Rettenmaier, R Snelling, W Bryks, J Banwell, WT Wipke, ... The Journal of Organic Chemistry 76 (23), 9602-9610, 2011 | 161 | 2011 |
| An expanded allosteric network in PTP1B by multitemperature crystallography, fragment screening, and covalent tethering DA Keedy, ZB Hill, JT Biel, E Kang, TJ Rettenmaier, J Brandao-Neto, ... Elife 7, e36307, 2018 | 157 | 2018 |
| A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1 TJ Rettenmaier, JD Sadowsky, ND Thomsen, SC Chen, AK Doak, ... Proceedings of the National Academy of Sciences 111 (52), 18590-18595, 2014 | 94 | 2014 |
| Cacidases: caspases can cleave after aspartate, glutamate and phosphoserine residues JE Seaman, O Julien, PS Lee, TJ Rettenmaier, ND Thomsen, JA Wells Cell Death & Differentiation 23 (10), 1717-1726, 2016 | 88 | 2016 |
| Kinase atlas: druggability analysis of potential allosteric sites in kinases C Yueh, J Rettenmaier, B Xia, DR Hall, A Alekseenko, KA Porter, ... Journal of medicinal chemistry 62 (14), 6512-6524, 2019 | 69 | 2019 |
| FP tethering: a screening technique to rapidly identify compounds that disrupt protein–protein interactions JM Lodge, TJ Rettenmaier, JA Wells, WC Pomerantz, AK Mapp MedChemComm 5 (3), 370-375, 2014 | 43 | 2014 |
| Identification of a covalent molecular inhibitor of anti-apoptotic BFL-1 by disulfide tethering EP Harvey, ZJ Hauseman, DT Cohen, TJ Rettenmaier, S Lee, AJ Huhn, ... Cell chemical biology 27 (6), 647-656. e6, 2020 | 35 | 2020 |
| Small-molecule allosteric modulators of the protein kinase PDK1 from structure-based docking TJ Rettenmaier, H Fan, J Karpiak, A Doak, A Sali, BK Shoichet, JA Wells Journal of medicinal chemistry 58 (20), 8285-8291, 2015 | 32 | 2015 |
| Redox priming promotes Aurora A activation during mitosis DC Lim, V Joukov, TJ Rettenmaier, A Kumagai, WG Dunphy, JA Wells, ... Science signaling 13 (641), eabb6707, 2020 | 23 | 2020 |
| An expanded allosteric network in PTP1B by multitemperature crystallography, fragment screening, and covalent tethering. Elife [Internet] DA Keedy, ZB Hill, JT Biel, E Kang, TJ Rettenmaier, J Brandão-Neto, ... DOI, 2018 | 8 | 2018 |
| Covalent inhibition of pro-apoptotic BAX MW McHenry, P Shi, CM Camara, DT Cohen, TJ Rettenmaier, U Adhikary, ... Nature Chemical Biology, 1-11, 2024 | 6 | 2024 |
| Site‐Directed Fragment Discovery for Allostery TJ Rettenmaier, SA Hudson, JA Wells Fragment‐based Drug Discovery Lessons and Outlook, 247-266, 2016 | 3 | 2016 |
| New routes for PTP1B allosteric inhibition by multitemperature crystallography, fragment screening and covalent tethering DA Keedy, ZB Hill, JT Biel, E Kang, TJ Rettenmaier, J Brandao-Neto, ... bioRxiv, 218966, 2017 | 2 | 2017 |
| Discovering and Manipulating Protein Conformational Heterogeneity and Function D Keedy, H van den Bedem, J Rettenmaier, J Wells, J Fraser Biophysical Journal 106 (2), 635a-636a, 2014 | | 2014 |
